GluK1 antagonists from 6-(carboxy)phenyl decahydroisoquinoline derivatives. SAR and evaluation of a prodrug strategy for oral efficacy in pain models

  1. Martinez-Perez, J.A.
  2. Iyengar, S.
  3. Shannon, H.E.
  4. Bleakman, D.
  5. Alt, A.
  6. Arnold, B.M.
  7. Bell, M.G.
  8. Bleisch, T.J.
  9. Castaño, A.M.
  10. Del Prado, M.
  11. Dominguez, E.
  12. Escribano, A.M.
  13. Filla, S.A.
  14. Ho, K.H.
  15. Hudziak, K.J.
  16. Jones, C.K.
  17. Mateo, A.
  18. Mathes, B.M.
  19. Mattiuz, E.L.
  20. Ogden, A.M.L.
  21. Simmons, R.M.A.
  22. Stack, D.R.
  23. Stratford, R.E.
  24. Winter, M.A.
  25. Wu, Z.
  26. Ornstein, P.L.
  27. Montrer des auteurs +
Revue:
Bioorganic and Medicinal Chemistry Letters

ISSN: 0960-894X 1464-3405

Année de publication: 2013

Volumen: 23

Número: 23

Pages: 6459-6462

Type: Article

DOI: 10.1016/J.BMCL.2013.09.046 GOOGLE SCHOLAR